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BioAssay: AID 162623

Inhibitory activity against porcine kidney prolidase

Inhibitory activity against porcine kidney prolidase ..more
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 Tested Compounds
 Tested Compounds
All(3)
 
 
Active(1)
 
 
Unspecified(2)
 
 
 Tested Substances
 Tested Substances
All(3)
 
 
Active(1)
 
 
Unspecified(2)
 
 
 Related BioAssays
 Related BioAssays
AID: 162623
Data Source: ChEMBL (159886)
BioAssay Type: Confirmatory, Concentration-Response Relationship Observed
Depositor Category: Literature, Extracted
BioAssay Version:
Deposit Date: 2010-05-20
Modify Date: 2014-08-23

Data Table ( Complete ):           View Active Data    View All Data
BioActive Compound: 1
Description:
Inhibitory activity against porcine kidney prolidase
Comment
Compounds with activity <= 50uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.
Putative Target:
ChEMBL Target ID: 11453
Target Type: SINGLE PROTEIN
Pref Name: Xaa-Pro dipeptidase
Synonyms: Imidodipeptidase;Peptidase D;Prolidase;Proline dipeptidase;X-Pro dipeptidase;Xaa-Pro dipeptidase;
Gene Name: PEPD;PRD;
Protein Accession: P12955;
Protein GI: 50403718;
Organism: Homo sapiens
Tax ID: 9606
Target Classification: enzyme protease metallo mg m24b
Confidence: Homologous single protein target assigned
Relationship Type: Homologous protein target assigned
Publication:
Journal: Bioorg. Med. Chem. Lett.
Year: 1995
Volume: 5
Issue: 23
First Page: 2825
Last Page: 2828
Categorized Comment - additional comments and annotations
From BioAssay Depositor:
Assay Type: Binding
Assay Data Source: Scientific Literature
Result Definitions
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TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1Ki*Ki PubChem standard valueFloatμM
3BEIBinding Efficiency Index(nM)Float
2SEISurface Efficiency Index(nM)Float
4LELigand EfficiencyFloat
5LLELipophilic Ligand EfficiencyFloat
6Ki activity commentKi activity commentString
7Ki standard flagKi standard flagInteger
8Ki qualifierKi qualifierString
9Ki published valueKi published valueFloatmM
10Ki standard valueKi standard valueFloatnM
11Ki data validityKi data validityString
12Ki activity commentKi activity commentString
13Ki standard flagKi standard flagInteger
14Ki qualifierKi qualifierString
15Ki published valueKi published valueFloatnM
16Ki standard valueKi standard valueFloatnM
17Ki data validityKi data validityString

* Activity Concentration.

Data Table (Concise)
Data Table ( Complete ):     View Active Data    View All Data
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