Kinase Inhibitor Selectivity Profiling Assay - BioAssay Summary
Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity are poorly defined, and an important step toward understanding the relationship between selectivity, efficacy and safety is the exploration of how inhibitors interact with the human kinome. We present interaction maps for 38 kinase inhibitors across more ..
 _
   
 Tested Compounds
 Tested Compounds
All(38)
 
 
Unspecified(38)
 
 
 Tested Substances
 Tested Substances
All(38)
 
 
Unspecified(38)
 
 
 Related BioAssays
 Related BioAssays
Table of Contents
AID: 1433
Data Source: Ambit Biosciences (Kinase inhibitor selectivity profiling)
BioAssay Type: Panel
BioAssay Version:
Deposit Date: 2008-11-19
Modify Date: 2008-11-21

Data Table (Complete):           All
Tested Compounds:
Description:
Helptop of page
Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity are poorly defined, and an important step toward understanding the relationship between selectivity, efficacy and safety is the exploration of how inhibitors interact with the human kinome. We present interaction maps for 38 kinase inhibitors across a panel of 317 kinases representing >50% of the predicted human protein kinome. The data constitute the most comprehensive study of kinase inhibitor selectivity to date and reveal a wide diversity of interaction patterns.
Panel Information
Helptop of page
Kinase inhibitor selectivity assay - Kinase inhibitor selectivity assay
    Data Table(All)Show more
PID§NameSubstancePanel TargetsDescription
ActiveInactive
1ABL1(T315I) Inhibition Activity218ABL1(T315I) [gi:62362414]
Inhibition Activity against kinase ABL1(T315I) is provided
2ALK Inhibition Activity15ALK [gi:29029632]
Inhibition Activity against kinase ALK is provided
3AURKA Inhibition Activity29AURKA [gi:38327562]
Inhibition Activity against kinase AURKA is provided
4AURKB Inhibition Activity211AURKB [gi:127796234]
Inhibition Activity against kinase AURKB is provided
5AURKC Inhibition Activity216AURKC [gi:3127068]
Inhibition Activity against kinase AURKC is provided
6AXL Inhibition Activity214AXL [gi:21536468]
Inhibition Activity against kinase AXL is provided
7BMPR2 Inhibition Activity6BMPR2 [gi:15451916]
Inhibition Activity against kinase BMPR2 is provided
8CDC2L1 Inhibition Activity7CDC2L1 [gi:16332362]
Inhibition Activity against kinase CDC2L1 is provided
9CDC2L2 Inhibition Activity7CDC2L2 [gi:148763347]
Inhibition Activity against kinase CDC2L2 is provided
10CDK11 Inhibition Activity110CDK11 [gi:30387611]
Inhibition Activity against kinase CDK11 is provided
11CDK7 Inhibition Activity111CDK7 [gi:4502743]
Inhibition Activity against kinase CDK7 is provided
12CDK8 Inhibition Activity17CDK8 [gi:4502745]
Inhibition Activity against kinase CDK8 is provided
13CDK9 Inhibition Activity15CDK9 [gi:4502747]
Inhibition Activity against kinase CDK9 is provided
14CLK1 Inhibition Activity16CLK1 [gi:632964]
Inhibition Activity against kinase CLK1 is provided
15CLK4 Inhibition Activity112CLK4 [gi:10190706]
Inhibition Activity against kinase CLK4 is provided
16CSF1R Inhibition Activity915CSF1R [gi:27262659]
Inhibition Activity against kinase CSF1R is provided
17DDR1 Inhibition Activity519DDR1 [gi:38327632]
Inhibition Activity against kinase DDR1 is provided
18DDR2 Inhibition Activity211DDR2 [gi:433338]
Inhibition Activity against kinase DDR2 is provided
19EGFR(G719C) Inhibition Activity713EGFR(G719C) [gi:29725609]
Inhibition Activity against kinase EGFR(G719C) is provided
20EPHA3 Inhibition Activity113EPHA3 [gi:21361241]
Inhibition Activity against kinase EPHA3 is provided
21EPHA6 Inhibition Activity16EPHA6 [gi:145312251]
Inhibition Activity against kinase EPHA6 is provided
22EPHA7 Inhibition Activity10EPHA7 [gi:4758282]
Inhibition Activity against kinase EPHA7 is provided
23EPHB3 Inhibition Activity12EPHB3 [gi:17975768]
Inhibition Activity against kinase EPHB3 is provided
24EPHB4 Inhibition Activity17EPHB4 [gi:32528301]
Inhibition Activity against kinase EPHB4 is provided
25ERK8 Inhibition Activity9ERK8 [gi:95147356]
Inhibition Activity against kinase ERK8 is provided
26FLT1 Inhibition Activity417FLT1 [gi:156104876]
Inhibition Activity against kinase FLT1 is provided
27FLT3 Inhibition Activity910FLT3 [gi:121114304]
Inhibition Activity against kinase FLT3 is provided
28FLT3(D835H) Inhibition Activity716FLT3(D835H) [gi:121114304]
Inhibition Activity against kinase FLT3(D835H) is provided
29FLT3(D835Y) Inhibition Activity417FLT3(D835Y) [gi:121114304]
Inhibition Activity against kinase FLT3(D835Y) is provided
30FLT3(ITD) Inhibition Activity613FLT3(ITD) [gi:121114304]
Inhibition Activity against kinase FLT3(ITD) is provided
31FLT3(N841I) Inhibition Activity814FLT3(N841I) [gi:121114304]
Inhibition Activity against kinase FLT3(N841I) is provided
32FLT4 Inhibition Activity117FLT4 [gi:297050]
Inhibition Activity against kinase FLT4 is provided
33FRK Inhibition Activity121FRK [gi:4503787]
Inhibition Activity against kinase FRK is provided
34INSRR Inhibition Activity6INSRR [gi:31657140]
Inhibition Activity against kinase INSRR is provided
35JNK2 Inhibition Activity14JNK2 [gi:21237739]
Inhibition Activity against kinase JNK2 is provided
36KIT Inhibition Activity1011KIT [gi:4557695]
Inhibition Activity against kinase KIT is provided
37KIT(D816V) Inhibition Activity320KIT(D816V) [gi:4557695]
Inhibition Activity against kinase KIT(D816V) is provided
38KIT(V559D T670I) Inhibition Activity613KIT(V559D T670I) [gi:4557695]
Inhibition Activity against kinase KIT(V559D T670I) is provided
39KIT(V559D V654A) Inhibition Activity415KIT(V559D V654A) [gi:4557695]
Inhibition Activity against kinase KIT(V559D V654A) is provided
40KIT(V559D) Inhibition Activity913KIT(V559D) [gi:4557695]
Inhibition Activity against kinase KIT(V559D) is provided
41LATS2 Inhibition Activity9LATS2 [gi:126507091]
Inhibition Activity against kinase LATS2 is provided
42LIMK2 Inhibition Activity7LIMK2 [gi:5031869]
Inhibition Activity against kinase LIMK2 is provided
43LOK Inhibition Activity222LOK [gi:4001688]
Inhibition Activity against kinase LOK is provided
44LTK Inhibition Activity12LTK [gi:46249416]
Inhibition Activity against kinase LTK is provided
45MAP4K1 Inhibition Activity113MAP4K1 [gi:110611908]
Inhibition Activity against kinase MAP4K1 is provided
46MAP4K3 Inhibition Activity114MAP4K3 [gi:15451902]
Inhibition Activity against kinase MAP4K3 is provided
47MAP4K5 Inhibition Activity117MAP4K5 [gi:14589909]
Inhibition Activity against kinase MAP4K5 is provided
48MERTK Inhibition Activity115MERTK [gi:505665]
Inhibition Activity against kinase MERTK is provided
49MET Inhibition Activity10MET [gi:42741655]
Inhibition Activity against kinase MET is provided
50MKNK1 Inhibition Activity9MKNK1 [gi:55957746]
Inhibition Activity against kinase MKNK1 is provided
51MKNK2 Inhibition Activity111MKNK2 [gi:6563264]
Inhibition Activity against kinase MKNK2 is provided
52MST1 Inhibition Activity18MST1 [gi:5454096]
Inhibition Activity against kinase MST1 is provided
53MST2 Inhibition Activity112MST2 [gi:103471999]
Inhibition Activity against kinase MST2 is provided
54MUSK Inhibition Activity28MUSK [gi:5031927]
Inhibition Activity against kinase MUSK is provided
55PDGFRA Inhibition Activity814PDGFRA [gi:5453870]
Inhibition Activity against kinase PDGFRA is provided
56PDGFRB Inhibition Activity1013PDGFRB [gi:4505683]
Inhibition Activity against kinase PDGFRB is provided
57PKAC-alpha Inhibition Activity6PKAC-alpha [gi:4506055]
Inhibition Activity against kinase PKAC-alpha is provided
58PLK3 Inhibition Activity3PLK3 [gi:41872374]
Inhibition Activity against kinase PLK3 is provided
59RET Inhibition Activity19RET [gi:10862701]
Inhibition Activity against kinase RET is provided
60RET(M918T) Inhibition Activity218RET(M918T) [gi:10862701]
Inhibition Activity against kinase RET(M918T) is provided
61RIPK1 Inhibition Activity8RIPK1 [gi:57242761]
Inhibition Activity against kinase RIPK1 is provided
62RPS6KA4(Kin.Dom.1 - N-terminal) Inhibition Activity10RPS6KA4(Kin.Dom.1 - N-terminal) [gi:55743138]
Inhibition Activity against kinase RPS6KA4(Kin.Dom.1 - N-terminal) is provided
63RPS6KA5(Kin.Dom.1 - N-terminal) Inhibition Activity8RPS6KA5(Kin.Dom.1 - N-terminal) [gi:32528297]
Inhibition Activity against kinase RPS6KA5(Kin.Dom.1 - N-terminal) is provided
64SLK Inhibition Activity121SLK [gi:41281453]
Inhibition Activity against kinase SLK is provided
65STK33 Inhibition Activity19STK33 [gi:23943882]
Inhibition Activity against kinase STK33 is provided
66TIE1 Inhibition Activity215TIE1 [gi:4885631]
Inhibition Activity against kinase TIE1 is provided
67TIE2 Inhibition Activity12TIE2 [gi:88758596]
Inhibition Activity against kinase TIE2 is provided
68TRKA Inhibition Activity111TRKA [gi:59889558]
Inhibition Activity against kinase TRKA is provided
69TRKB Inhibition Activity111TRKB [gi:21361306]
Inhibition Activity against kinase TRKB is provided
70TRKC Inhibition Activity12TRKC [gi:442390]
Inhibition Activity against kinase TRKC is provided
71VEGFR2 Inhibition Activity314VEGFR2 [gi:11321597]
Inhibition Activity against kinase VEGFR2 is provided
72YANK2 Inhibition Activity5YANK2 [gi:8923754]
Inhibition Activity against kinase YANK2 is provided
73ABL1 Inhibition Activity218ABL1 [gi:62362414]
Inhibition Activity against kinase ABL1 is provided
74BLK Inhibition Activity119BLK [gi:33469982]
Inhibition Activity against kinase BLK is provided
75BRAF Inhibition Activity10BRAF [gi:33188459]
Inhibition Activity against kinase BRAF is provided
76BRAF(V600E) Inhibition Activity10BRAF(V600E) [gi:33188459]
Inhibition Activity against kinase BRAF(V600E) is provided
77CIT Inhibition Activity20CIT [gi:32698688]
Inhibition Activity against kinase CIT is provided
78EGFR Inhibition Activity611EGFR [gi:29725609]
Inhibition Activity against kinase EGFR is provided
79EGFR(G719S) Inhibition Activity611EGFR(G719S) [gi:29725609]
Inhibition Activity against kinase EGFR(G719S) is provided
80EGFR(L747-E749del A750P) Inhibition Activity514EGFR(L747-E749del A750P) [gi:29725609]
Inhibition Activity against kinase EGFR(L747-E749del A750P) is provided
81EGFR(L747-S752del P753S) Inhibition Activity611EGFR(L747-S752del P753S) [gi:29725609]
Inhibition Activity against kinase EGFR(L747-S752del P753S) is provided
82EGFR(L747-T751del Sins) Inhibition Activity611EGFR(L747-T751del Sins) [gi:29725609]
Inhibition Activity against kinase EGFR(L747-T751del Sins) is provided
83EGFR(L861Q) Inhibition Activity511EGFR(L861Q) [gi:29725609]
Inhibition Activity against kinase EGFR(L861Q) is provided
84FGFR1 Inhibition Activity16FGFR1 [gi:13186234]
Inhibition Activity against kinase FGFR1 is provided
85FGFR4 Inhibition Activity6FGFR4 [gi:47524177]
Inhibition Activity against kinase FGFR4 is provided
86FGR Inhibition Activity117FGR [gi:4885235]
Inhibition Activity against kinase FGR is provided
87FYN Inhibition Activity115FYN [gi:23510362]
Inhibition Activity against kinase FYN is provided
88GCN2(Kin.Dom.2 S808G) Inhibition Activity12GCN2(Kin.Dom.2 S808G) [gi:65287717]
Inhibition Activity against kinase GCN2(Kin.Dom.2 S808G) is provided
89LCK Inhibition Activity123LCK [gi:112789546]
Inhibition Activity against kinase LCK is provided
90LYN Inhibition Activity120LYN [gi:4505055]
Inhibition Activity against kinase LYN is provided
91PTK6 Inhibition Activity19PTK6 [gi:5174647]
Inhibition Activity against kinase PTK6 is provided
92RAF1 Inhibition Activity10RAF1 [gi:4506401]
Inhibition Activity against kinase RAF1 is provided
93TNNI3K Inhibition Activity14TNNI3K [gi:7705748]
Inhibition Activity against kinase TNNI3K is provided
94ZAK Inhibition Activity311ZAK [gi:19526767]
Inhibition Activity against kinase ZAK is provided
95ABL1(E255K) Inhibition Activity114ABL1(E255K) [gi:62362414]
Inhibition Activity against kinase ABL1(E255K) is provided
96ABL1(H396P) Inhibition Activity215ABL1(H396P) [gi:62362414]
Inhibition Activity against kinase ABL1(H396P) is provided
97ABL1(M351T) Inhibition Activity414ABL1(M351T) [gi:62362414]
Inhibition Activity against kinase ABL1(M351T) is provided
98ABL1(Q252H) Inhibition Activity216ABL1(Q252H) [gi:62362414]
Inhibition Activity against kinase ABL1(Q252H) is provided
99ABL1(Y253F) Inhibition Activity216ABL1(Y253F) [gi:62362414]
Inhibition Activity against kinase ABL1(Y253F) is provided
100ABL2 Inhibition Activity411ABL2 [gi:153266757]
Inhibition Activity against kinase ABL2 is provided
101AMPK-alpha1 Inhibition Activity18AMPK-alpha1 [gi:4115829]
Inhibition Activity against kinase AMPK-alpha1 is provided
102ANKK1 Inhibition Activity9ANKK1 [gi:30425444]
Inhibition Activity against kinase ANKK1 is provided
103CAMK1 Inhibition Activity7CAMK1 [gi:4502553]
Inhibition Activity against kinase CAMK1 is provided
104CAMK4 Inhibition Activity5CAMK4 [gi:4502557]
Inhibition Activity against kinase CAMK4 is provided
105CAMKK1 Inhibition Activity19CAMKK1 [gi:14150045]
Inhibition Activity against kinase CAMKK1 is provided
106CAMKK2 Inhibition Activity18CAMKK2 [gi:27437015]
Inhibition Activity against kinase CAMKK2 is provided
107CDK2 Inhibition Activity15CDK2 [gi:16936528]
Inhibition Activity against kinase CDK2 is provided
108CDK3 Inhibition Activity5CDK3 [gi:4557439]
Inhibition Activity against kinase CDK3 is provided
109CDK5 Inhibition Activity7CDK5 [gi:4826675]
Inhibition Activity against kinase CDK5 is provided
110CLK2 Inhibition Activity112CLK2 [gi:47717134]
Inhibition Activity against kinase CLK2 is provided
111CSK Inhibition Activity18CSK [gi:4758078]
Inhibition Activity against kinase CSK is provided
112CSNK1D Inhibition Activity11CSNK1D [gi:20544145]
Inhibition Activity against kinase CSNK1D is provided
113CSNK1E Inhibition Activity14CSNK1E [gi:4503093]
Inhibition Activity against kinase CSNK1E is provided
114CSNK1G2 Inhibition Activity5CSNK1G2 [gi:153791733]
Inhibition Activity against kinase CSNK1G2 is provided
115CSNK1G3 Inhibition Activity5CSNK1G3 [gi:73532778]
Inhibition Activity against kinase CSNK1G3 is provided
116DAPK3 Inhibition Activity16DAPK3 [gi:4557511]
Inhibition Activity against kinase DAPK3 is provided
117DLK Inhibition Activity8DLK [gi:21735552]
Inhibition Activity against kinase DLK is provided
118EGFR(E746-A750del) Inhibition Activity68EGFR(E746-A750del) [gi:29725609]
Inhibition Activity against kinase EGFR(E746-A750del) is provided
119EGFR(L858R) Inhibition Activity610EGFR(L858R) [gi:29725609]
Inhibition Activity against kinase EGFR(L858R) is provided
120EPHA2 Inhibition Activity19EPHA2 [gi:32967311]
Inhibition Activity against kinase EPHA2 is provided
121EPHA4 Inhibition Activity18EPHA4 [gi:4758280]
Inhibition Activity against kinase EPHA4 is provided
122EPHA5 Inhibition Activity16EPHA5 [gi:56119209]
Inhibition Activity against kinase EPHA5 is provided
123EPHA8 Inhibition Activity112EPHA8 [gi:10140845]
Inhibition Activity against kinase EPHA8 is provided
124EPHB1 Inhibition Activity18EPHB1 [gi:4758284]
Inhibition Activity against kinase EPHB1 is provided
125EPHB2 Inhibition Activity16EPHB2 [gi:111118978]
Inhibition Activity against kinase EPHB2 is provided
126FER Inhibition Activity8FER [gi:119964721]
Inhibition Activity against kinase FER is provided
127FES Inhibition Activity4FES [gi:4503687]
Inhibition Activity against kinase FES is provided
128FGFR2 Inhibition Activity13FGFR2 [gi:189083817]
Inhibition Activity against kinase FGFR2 is provided
129GAK Inhibition Activity318GAK [gi:157384971]
Inhibition Activity against kinase GAK is provided
130HCK Inhibition Activity114HCK [gi:30795229]
Inhibition Activity against kinase HCK is provided
131ITK Inhibition Activity8ITK [gi:15718680]
Inhibition Activity against kinase ITK is provided
132JAK2(Kin.Dom.2/JH1 - catalytic) Inhibition Activity19JAK2(Kin.Dom.2/JH1 - catalytic) [gi:4826776]
Inhibition Activity against kinase JAK2(Kin.Dom.2/JH1 - catalytic) is provided
133JAK3(Kin.Dom.2/JH1 - catalytic) Inhibition Activity212JAK3(Kin.Dom.2/JH1 - catalytic) [gi:47157315]
Inhibition Activity against kinase JAK3(Kin.Dom.2/JH1 - catalytic) is provided
134JNK1 Inhibition Activity7JNK1 [gi:4506095]
Inhibition Activity against kinase JNK1 is provided
135JNK3 Inhibition Activity13JNK3 [gi:4506081]
Inhibition Activity against kinase JNK3 is provided
136LATS1 Inhibition Activity8LATS1 [gi:4758666]
Inhibition Activity against kinase LATS1 is provided
137MAP4K4 Inhibition Activity14MAP4K4 [gi:22035604]
Inhibition Activity against kinase MAP4K4 is provided
138MELK Inhibition Activity9MELK [gi:7661974]
Inhibition Activity against kinase MELK is provided
139MYLK2 Inhibition Activity11MYLK2 [gi:14993776]
Inhibition Activity against kinase MYLK2 is provided
140MYO3A Inhibition Activity2MYO3A [gi:145275208]
Inhibition Activity against kinase MYO3A is provided
141MYO3B Inhibition Activity3MYO3B [gi:134288892]
Inhibition Activity against kinase MYO3B is provided
142NEK5 Inhibition Activity5NEK5 [gi:83627721]
Inhibition Activity against kinase NEK5 is provided
143NLK Inhibition Activity8NLK [gi:149408126]
Inhibition Activity against kinase NLK is provided
144PCTK1 Inhibition Activity111PCTK1 [gi:5453860]
Inhibition Activity against kinase PCTK1 is provided
145PCTK2 Inhibition Activity8PCTK2 [gi:36617]
Inhibition Activity against kinase PCTK2 is provided
146PCTK3 Inhibition Activity6PCTK3 [gi:47078229]
Inhibition Activity against kinase PCTK3 is provided
147PFTK1 Inhibition Activity7PFTK1 [gi:6912584]
Inhibition Activity against kinase PFTK1 is provided
148PKAC-beta Inhibition Activity5PKAC-beta [gi:4506057]
Inhibition Activity against kinase PKAC-beta is provided
149PRKCQ Inhibition Activity27PRKCQ [gi:5453976]
Inhibition Activity against kinase PRKCQ is provided
150PRKD1 Inhibition Activity7PRKD1 [gi:115529463]
Inhibition Activity against kinase PRKD1 is provided
151PRKD2 Inhibition Activity8PRKD2 [gi:19923468]
Inhibition Activity against kinase PRKD2 is provided
152PRKD3 Inhibition Activity8PRKD3 [gi:5031689]
Inhibition Activity against kinase PRKD3 is provided
153PRKR Inhibition Activity12PRKR [gi:4506103]
Inhibition Activity against kinase PRKR is provided
154PTK2B Inhibition Activity17PTK2B [gi:27886588]
Inhibition Activity against kinase PTK2B is provided
155RIPK2 Inhibition Activity114RIPK2 [gi:4506537]
Inhibition Activity against kinase RIPK2 is provided
156ROS1 Inhibition Activity6ROS1 [gi:19924165]
Inhibition Activity against kinase ROS1 is provided
157RPS6KA2(Kin.Dom.2 - C-terminal) Inhibition Activity7RPS6KA2(Kin.Dom.2 - C-terminal) [gi:55743136]
Inhibition Activity against kinase RPS6KA2(Kin.Dom.2 - C-terminal) is provided
158RPS6KA6(Kin.Dom.2 - C-terminal) Inhibition Activity8RPS6KA6(Kin.Dom.2 - C-terminal) [gi:7657526]
Inhibition Activity against kinase RPS6KA6(Kin.Dom.2 - C-terminal) is provided
159SNF1LK Inhibition Activity29SNF1LK [gi:116256471]
Inhibition Activity against kinase SNF1LK is provided
160SRC Inhibition Activity117SRC [gi:4885609]
Inhibition Activity against kinase SRC is provided
161SRMS Inhibition Activity10SRMS [gi:18250298]
Inhibition Activity against kinase SRMS is provided
162STK36 Inhibition Activity11STK36 [gi:24308123]
Inhibition Activity against kinase STK36 is provided
163SYK Inhibition Activity7SYK [gi:21361553]
Inhibition Activity against kinase SYK is provided
164TESK1 Inhibition Activity7TESK1 [gi:66932999]
Inhibition Activity against kinase TESK1 is provided
165TGFBR2 Inhibition Activity6TGFBR2 [gi:67782324]
Inhibition Activity against kinase TGFBR2 is provided
166TNIK Inhibition Activity114TNIK [gi:55741807]
Inhibition Activity against kinase TNIK is provided
167TNK1 Inhibition Activity110TNK1 [gi:23273502]
Inhibition Activity against kinase TNK1 is provided
168TTK Inhibition Activity13TTK [gi:23308722]
Inhibition Activity against kinase TTK is provided
169TYK2(Kin.Dom.2/JH1 - catalytic) Inhibition Activity7TYK2(Kin.Dom.2/JH1 - catalytic) [gi:37504]
Inhibition Activity against kinase TYK2(Kin.Dom.2/JH1 - catalytic) is provided
170YES Inhibition Activity117YES [gi:4885661]
Inhibition Activity against kinase YES is provided
171YSK1 Inhibition Activity9YSK1 [gi:21361358]
Inhibition Activity against kinase YSK1 is provided
172p38-alpha Inhibition Activity34p38-alpha [gi:20986512]
Inhibition Activity against kinase p38-alpha is provided
173p38-beta Inhibition Activity7p38-beta [gi:20128774]
Inhibition Activity against kinase p38-beta is provided
174p38-gamma Inhibition Activity6p38-gamma [gi:1772646]
Inhibition Activity against kinase p38-gamma is provided
175EGFR(S752-I759del) Inhibition Activity510EGFR(S752-I759del) [gi:29725609]
Inhibition Activity against kinase EGFR(S752-I759del) is provided
176ERBB2 Inhibition Activity17ERBB2 [gi:54792098]
Inhibition Activity against kinase ERBB2 is provided
177ERBB4 Inhibition Activity12ERBB4 [gi:110825958]
Inhibition Activity against kinase ERBB4 is provided
178MEK2 Inhibition Activity13MEK2 [gi:13489054]
Inhibition Activity against kinase MEK2 is provided
179PLK4 Inhibition Activity211PLK4 [gi:16215696]
Inhibition Activity against kinase PLK4 is provided
180DMPK2 Inhibition Activity7DMPK2 [gi:156766068]
Inhibition Activity against kinase DMPK2 is provided
181EPHA1 Inhibition Activity18EPHA1 [gi:56119207]
Inhibition Activity against kinase EPHA1 is provided
182MRCKA Inhibition Activity7MRCKA [gi:30089962]
Inhibition Activity against kinase MRCKA is provided
183MRCKB Inhibition Activity7MRCKB [gi:115527097]
Inhibition Activity against kinase MRCKB is provided
184PTK2 Inhibition Activity4PTK2 [gi:24476013]
Inhibition Activity against kinase PTK2 is provided
185DCAMKL1 Inhibition Activity6DCAMKL1 [gi:4758128]
Inhibition Activity against kinase DCAMKL1 is provided
186DCAMKL2 Inhibition Activity4DCAMKL2 [gi:156713430]
Inhibition Activity against kinase DCAMKL2 is provided
187DCAMKL3 Inhibition Activity19DCAMKL3 [gi:113414461]
Inhibition Activity against kinase DCAMKL3 is provided
188DRAK1 Inhibition Activity110DRAK1 [gi:109255245]
Inhibition Activity against kinase DRAK1 is provided
189DYRK1B Inhibition Activity9DYRK1B [gi:4758222]
Inhibition Activity against kinase DYRK1B is provided
190ERK3 Inhibition Activity5ERK3 [gi:4506091]
Inhibition Activity against kinase ERK3 is provided
191ERK4 Inhibition Activity4ERK4 [gi:89276769]
Inhibition Activity against kinase ERK4 is provided
192ERK5 Inhibition Activity4ERK5 [gi:20986497]
Inhibition Activity against kinase ERK5 is provided
193GSK3A Inhibition Activity5GSK3A [gi:49574532]
Inhibition Activity against kinase GSK3A is provided
194GSK3B Inhibition Activity9GSK3B [gi:21361340]
Inhibition Activity against kinase GSK3B is provided
195IRAK3 Inhibition Activity12IRAK3 [gi:6005792]
Inhibition Activity against kinase IRAK3 is provided
196MLCK Inhibition Activity15MLCK [gi:146219832]
Inhibition Activity against kinase MLCK is provided
197PAK3 Inhibition Activity17PAK3 [gi:4505601]
Inhibition Activity against kinase PAK3 is provided
198PHKG1 Inhibition Activity210PHKG1 [gi:5453882]
Inhibition Activity against kinase PHKG1 is provided
199SNARK Inhibition Activity111SNARK [gi:13569922]
Inhibition Activity against kinase SNARK is provided
200AAK1 Inhibition Activity111AAK1 [gi:148277037]
Inhibition Activity against kinase AAK1 is provided
201AMPK-alpha2 Inhibition Activity7AMPK-alpha2 [gi:46877068]
Inhibition Activity against kinase AMPK-alpha2 is provided
202ARK5 Inhibition Activity17ARK5 [gi:7662170]
Inhibition Activity against kinase ARK5 is provided
203BIKE Inhibition Activity210BIKE [gi:38787904]
Inhibition Activity against kinase BIKE is provided
204CHEK1 Inhibition Activity16CHEK1 [gi:166295192]
Inhibition Activity against kinase CHEK1 is provided
205CSNK2A1 Inhibition Activity7CSNK2A1 [gi:4503095]
Inhibition Activity against kinase CSNK2A1 is provided
206CSNK2A2 Inhibition Activity16CSNK2A2 [gi:4503097]
Inhibition Activity against kinase CSNK2A2 is provided
207DRAK2 Inhibition Activity18DRAK2 [gi:4758194]
Inhibition Activity against kinase DRAK2 is provided
208FGFR3 Inhibition Activity10FGFR3 [gi:4503711]
Inhibition Activity against kinase FGFR3 is provided
209FGFR3(G697C) Inhibition Activity10FGFR3(G697C) [gi:4503711]
Inhibition Activity against kinase FGFR3(G697C) is provided
210IKK-epsilon Inhibition Activity17IKK-epsilon [gi:7661946]
Inhibition Activity against kinase IKK-epsilon is provided
211JAK1(Kin.Dom.1/JH2 - pseudokinase) Inhibition Activity4JAK1(Kin.Dom.1/JH2 - pseudokinase) [gi:102469034]
Inhibition Activity against kinase JAK1(Kin.Dom.1/JH2 - pseudokinase) is provided
212LKB1 Inhibition Activity6LKB1 [gi:4507271]
Inhibition Activity against kinase LKB1 is provided
213MAP3K4 Inhibition Activity6MAP3K4 [gi:55956904]
Inhibition Activity against kinase MAP3K4 is provided
214MARK1 Inhibition Activity17MARK1 [gi:55665540]
Inhibition Activity against kinase MARK1 is provided
215MARK2 Inhibition Activity16MARK2 [gi:86990441]
Inhibition Activity against kinase MARK2 is provided
216MARK3 Inhibition Activity17MARK3 [gi:46852166]
Inhibition Activity against kinase MARK3 is provided
217MARK4 Inhibition Activity16MARK4 [gi:33636756]
Inhibition Activity against kinase MARK4 is provided
218MEK1 Inhibition Activity10MEK1 [gi:5579478]
Inhibition Activity against kinase MEK1 is provided
219MLK1 Inhibition Activity19MLK1 [gi:52421790]
Inhibition Activity against kinase MLK1 is provided
220MLK3 Inhibition Activity7MLK3 [gi:4505195]
Inhibition Activity against kinase MLK3 is provided
221MST3 Inhibition Activity7MST3 [gi:20070158]
Inhibition Activity against kinase MST3 is provided
222MST4 Inhibition Activity6MST4 [gi:15011880]
Inhibition Activity against kinase MST4 is provided
223MYLK Inhibition Activity8MYLK [gi:116008188]
Inhibition Activity against kinase MYLK is provided
224NEK2 Inhibition Activity6NEK2 [gi:4505373]
Inhibition Activity against kinase NEK2 is provided
225NEK6 Inhibition Activity1NEK6 [gi:19923407]
Inhibition Activity against kinase NEK6 is provided
226NEK7 Inhibition Activity4NEK7 [gi:19424132]
Inhibition Activity against kinase NEK7 is provided
227NEK9 Inhibition Activity2NEK9 [gi:31543286]
Inhibition Activity against kinase NEK9 is provided
228PHKG2 Inhibition Activity24PHKG2 [gi:4505785]
Inhibition Activity against kinase PHKG2 is provided
229PIP5K1A Inhibition Activity8PIP5K1A [gi:1743873]
Inhibition Activity against kinase PIP5K1A is provided
230PIP5K2B Inhibition Activity9PIP5K2B [gi:4505819]
Inhibition Activity against kinase PIP5K2B is provided
231PKN1 Inhibition Activity27PKN1 [gi:47132591]
Inhibition Activity against kinase PKN1 is provided
232PKN2 Inhibition Activity16PKN2 [gi:5453974]
Inhibition Activity against kinase PKN2 is provided
233RIOK1 Inhibition Activity8RIOK1 [gi:23510356]
Inhibition Activity against kinase RIOK1 is provided
234RIOK3 Inhibition Activity7RIOK3 [gi:22325377]
Inhibition Activity against kinase RIOK3 is provided
235RPS6KA1(Kin.Dom.1 - N-terminal) Inhibition Activity8RPS6KA1(Kin.Dom.1 - N-terminal) [gi:20149547]
Inhibition Activity against kinase RPS6KA1(Kin.Dom.1 - N-terminal) is provided
236RPS6KA2(Kin.Dom.1 - N-terminal) Inhibition Activity17RPS6KA2(Kin.Dom.1 - N-terminal) [gi:19923570]
Inhibition Activity against kinase RPS6KA2(Kin.Dom.1 - N-terminal) is provided
237RPS6KA3(Kin.Dom.1 - N-terminal) Inhibition Activity7RPS6KA3(Kin.Dom.1 - N-terminal) [gi:4759050]
Inhibition Activity against kinase RPS6KA3(Kin.Dom.1 - N-terminal) is provided
238RPS6KA6(Kin.Dom.1 - N-terminal) Inhibition Activity6RPS6KA6(Kin.Dom.1 - N-terminal) [gi:7657526]
Inhibition Activity against kinase RPS6KA6(Kin.Dom.1 - N-terminal) is provided
239SNF1LK2 Inhibition Activity211SNF1LK2 [gi:38569460]
Inhibition Activity against kinase SNF1LK2 is provided
240SRPK1 Inhibition Activity16SRPK1 [gi:47419936]
Inhibition Activity against kinase SRPK1 is provided
241SRPK2 Inhibition Activity6SRPK2 [gi:1857944]
Inhibition Activity against kinase SRPK2 is provided
242SgK085 Inhibition Activity6SgK085 [gi:167466233]
Inhibition Activity against kinase SgK085 is provided
243TLK2 Inhibition Activity5TLK2 [gi:6063019]
Inhibition Activity against kinase TLK2 is provided
244TYRO3 Inhibition Activity9TYRO3 [gi:27597078]
Inhibition Activity against kinase TYRO3 is provided
245WEE1 Inhibition Activity7WEE1 [gi:4507917]
Inhibition Activity against kinase WEE1 is provided
246ACVR1 Inhibition Activity8ACVR1 [gi:4501895]
Inhibition Activity against kinase ACVR1 is provided
247ADCK3 Inhibition Activity5ADCK3 [gi:34147522]
Inhibition Activity against kinase ADCK3 is provided
248ADCK4 Inhibition Activity6ADCK4 [gi:27363457]
Inhibition Activity against kinase ADCK4 is provided
249BMX Inhibition Activity16BMX [gi:4502435]
Inhibition Activity against kinase BMX is provided
250BTK Inhibition Activity15BTK [gi:4557377]
Inhibition Activity against kinase BTK is provided
251RPS6KA1(Kin.Dom.2 - C-terminal) Inhibition Activity9RPS6KA1(Kin.Dom.2 - C-terminal) [gi:20149547]
Inhibition Activity against kinase RPS6KA1(Kin.Dom.2 - C-terminal) is provided
252TEC Inhibition Activity5TEC [gi:130977759]
Inhibition Activity against kinase TEC is provided
253TGFBR1 Inhibition Activity5TGFBR1 [gi:4759226]
Inhibition Activity against kinase TGFBR1 is provided
254TXK Inhibition Activity18TXK [gi:148596974]
Inhibition Activity against kinase TXK is provided
255ACVR1B Inhibition Activity5ACVR1B [gi:4757720]
Inhibition Activity against kinase ACVR1B is provided
256ACVR2A Inhibition Activity2ACVR2A [gi:4501897]
Inhibition Activity against kinase ACVR2A is provided
257ACVR2B Inhibition Activity6ACVR2B [gi:116734708]
Inhibition Activity against kinase ACVR2B is provided
258ACVRL1 Inhibition Activity3ACVRL1 [gi:116734712]
Inhibition Activity against kinase ACVRL1 is provided
259DMPK Inhibition Activity18DMPK [gi:47059024]
Inhibition Activity against kinase DMPK is provided
260LIMK1 Inhibition Activity6LIMK1 [gi:4505001]
Inhibition Activity against kinase LIMK1 is provided
261PKMYT1 Inhibition Activity2PKMYT1 [gi:33383239]
Inhibition Activity against kinase PKMYT1 is provided
262TNK2 Inhibition Activity16TNK2 [gi:58331191]
Inhibition Activity against kinase TNK2 is provided
263CAMK1D Inhibition Activity15CAMK1D [gi:9966875]
Inhibition Activity against kinase CAMK1D is provided
264CLK3 Inhibition Activity5CLK3 [gi:153791372]
Inhibition Activity against kinase CLK3 is provided
265CSNK1A1L Inhibition Activity7CSNK1A1L [gi:21624639]
Inhibition Activity against kinase CSNK1A1L is provided
266NEK1 Inhibition Activity2NEK1 [gi:41872673]
Inhibition Activity against kinase NEK1 is provided
267PAK1 Inhibition Activity13PAK1 [gi:42794769]
Inhibition Activity against kinase PAK1 is provided
268PRKCD Inhibition Activity24PRKCD [gi:31377782]
Inhibition Activity against kinase PRKCD is provided
269RPS6KA4(Kin.Dom.2 - C-terminal) Inhibition Activity4RPS6KA4(Kin.Dom.2 - C-terminal) [gi:4506735]
Inhibition Activity against kinase RPS6KA4(Kin.Dom.2 - C-terminal) is provided
270CAMK2A Inhibition Activity15CAMK2A [gi:25952118]
Inhibition Activity against kinase CAMK2A is provided
271MLK2 Inhibition Activity5MLK2 [gi:21735550]
Inhibition Activity against kinase MLK2 is provided
272PIM1 Inhibition Activity13PIM1 [gi:4505811]
Inhibition Activity against kinase PIM1 is provided
273PIM2 Inhibition Activity12PIM2 [gi:42821112]
Inhibition Activity against kinase PIM2 is provided
274PIM3 Inhibition Activity16PIM3 [gi:49258202]
Inhibition Activity against kinase PIM3 is provided
275PRKCE Inhibition Activity13PRKCE [gi:4885563]
Inhibition Activity against kinase PRKCE is provided
276PRKCH Inhibition Activity13PRKCH [gi:28557781]
Inhibition Activity against kinase PRKCH is provided
277CAMK1G Inhibition Activity5CAMK1G [gi:14196445]
Inhibition Activity against kinase CAMK1G is provided
278MEK4 Inhibition Activity6MEK4 [gi:4506889]
Inhibition Activity against kinase MEK4 is provided
279MEK6 Inhibition Activity14MEK6 [gi:14589900]
Inhibition Activity against kinase MEK6 is provided
280STK16 Inhibition Activity7STK16 [gi:3367705]
Inhibition Activity against kinase STK16 is provided
281BRSK1 Inhibition Activity5BRSK1 [gi:24308326]
Inhibition Activity against kinase BRSK1 is provided
282BRSK2 Inhibition Activity14BRSK2 [gi:116089335]
Inhibition Activity against kinase BRSK2 is provided
283CSNK1G1 Inhibition Activity3CSNK1G1 [gi:98986450]
Inhibition Activity against kinase CSNK1G1 is provided
284MEK3 Inhibition Activity12MEK3 [gi:21618347]
Inhibition Activity against kinase MEK3 is provided
285PAK4 Inhibition Activity13PAK4 [gi:62422559]
Inhibition Activity against kinase PAK4 is provided
286PAK6 Inhibition Activity12PAK6 [gi:9910476]
Inhibition Activity against kinase PAK6 is provided
287PAK7/PAK5 Inhibition Activity13PAK7/PAK5 [gi:24308191]
Inhibition Activity against kinase PAK7/PAK5 is provided
288PDPK1 Inhibition Activity15PDPK1 [gi:4505695]
Inhibition Activity against kinase PDPK1 is provided
289PLK1 Inhibition Activity2PLK1 [gi:21359873]
Inhibition Activity against kinase PLK1 is provided
290TLK1 Inhibition Activity4TLK1 [gi:33636698]
Inhibition Activity against kinase TLK1 is provided
291AKT3 Inhibition Activity2AKT3 [gi:4885549]
Inhibition Activity against kinase AKT3 is provided
292CAMK2D Inhibition Activity14CAMK2D [gi:4426595]
Inhibition Activity against kinase CAMK2D is provided
293CAMK2G Inhibition Activity14CAMK2G [gi:26667211]
Inhibition Activity against kinase CAMK2G is provided
294DAPK1 Inhibition Activity15DAPK1 [gi:89363047]
Inhibition Activity against kinase DAPK1 is provided
295PRKG2 Inhibition Activity3PRKG2 [gi:5453978]
Inhibition Activity against kinase PRKG2 is provided
296DAPK2 Inhibition Activity14DAPK2 [gi:14670383]
Inhibition Activity against kinase DAPK2 is provided
297PIK3CA Inhibition Activity1PIK3CA [gi:54792082]
Inhibition Activity against kinase PIK3CA is provided
298PIK3CA(E545K) Inhibition Activity1PIK3CA(E545K) [gi:54792082]
Inhibition Activity against kinase PIK3CA(E545K) is provided
299AKT1 Inhibition Activity2AKT1 [gi:62241011]
Inhibition Activity against kinase AKT1 is provided
300AKT2 Inhibition Activity3AKT2 [gi:4502023]
Inhibition Activity against kinase AKT2 is provided
301CAMK2B Inhibition Activity13CAMK2B [gi:26051204]
Inhibition Activity against kinase CAMK2B is provided
302PAK2 Inhibition Activity12PAK2 [gi:32483399]
Inhibition Activity against kinase PAK2 is provided
303PRKG1 Inhibition Activity2PRKG1 [gi:10835242]
Inhibition Activity against kinase PRKG1 is provided
304PRKX Inhibition Activity2PRKX [gi:4826948]
Inhibition Activity against kinase PRKX is provided
305TSSK1 Inhibition Activity3TSSK1 [gi:14042947]
Inhibition Activity against kinase TSSK1 is provided
306ZAP70 Inhibition Activity2ZAP70 [gi:46488944]
Inhibition Activity against kinase ZAP70 is provided
307INSR Inhibition Activity4INSR [gi:119395736]
Inhibition Activity against kinase INSR is provided
308NDR2 Inhibition Activity3NDR2 [gi:24307971]
Inhibition Activity against kinase NDR2 is provided
309RPS6KA5(Kin.Dom.2 - C-terminal) Inhibition Activity3RPS6KA5(Kin.Dom.2 - C-terminal) [gi:32528295]
Inhibition Activity against kinase RPS6KA5(Kin.Dom.2 - C-terminal) is provided
310BMPR1A Inhibition Activity1BMPR1A [gi:41349437]
Inhibition Activity against kinase BMPR1A is provided
311ERK1 Inhibition Activity1ERK1 [gi:91718899]
Inhibition Activity against kinase ERK1 is provided
312ERK2 Inhibition Activity1ERK2 [gi:20986531]
Inhibition Activity against kinase ERK2 is provided
313IGF1R Inhibition Activity3IGF1R [gi:4557665]
Inhibition Activity against kinase IGF1R is provided
314MAP3K5 Inhibition Activity1MAP3K5 [gi:5174547]
Inhibition Activity against kinase MAP3K5 is provided
315MAPKAPK2 Inhibition Activity1MAPKAPK2 [gi:32481209]
Inhibition Activity against kinase MAPKAPK2 is provided
316YANK3 Inhibition Activity1YANK3 [gi:32455269]
Inhibition Activity against kinase YANK3 is provided
§ Panel component ID.
Comment
Helptop of page
Compounds with Kd equal or less than 10 uM are considered active.
Result Definitions
Helptop of page
Show more
TIDNameDescriptionPID§Panel TargetsHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1Outcome(ABL1(T315I))1ABL1(T315I)Outcome
2Kd(ABL1(T315I))*1FloatμM
3Outcome(ALK)2ALKOutcome
4Kd(ALK)*2FloatμM
5Outcome(AURKA)3AURKAOutcome
6Kd(AURKA)*3FloatμM
7Outcome(AURKB)4AURKBOutcome
8Kd(AURKB)*4FloatμM
9Outcome(AURKC)5AURKCOutcome
10Kd(AURKC)*5FloatμM
11Outcome(AXL)6AXLOutcome
12Kd(AXL)*6FloatμM
13Outcome(BMPR2)7BMPR2Outcome
14Kd(BMPR2)*7FloatμM
15Outcome(CDC2L1)8CDC2L1Outcome
16Kd(CDC2L1)*8FloatμM
17Outcome(CDC2L2)9CDC2L2Outcome
18Kd(CDC2L2)*9FloatμM
19Outcome(CDK11)10CDK11Outcome
20Kd(CDK11)*10FloatμM
21Outcome(CDK7)11CDK7Outcome
22Kd(CDK7)*11FloatμM
23Outcome(CDK8)12CDK8Outcome
24Kd(CDK8)*12FloatμM
25Outcome(CDK9)13CDK9Outcome
26Kd(CDK9)*13FloatμM
27Outcome(CLK1)14CLK1Outcome
28Kd(CLK1)*14FloatμM
29Outcome(CLK4)15CLK4Outcome
30Kd(CLK4)*15FloatμM
31Outcome(CSF1R)16CSF1ROutcome
32Kd(CSF1R)*16FloatμM
33Outcome(DDR1)17DDR1Outcome
34Kd(DDR1)*17FloatμM
35Outcome(DDR2)18DDR2Outcome
36Kd(DDR2)*18FloatμM
37Outcome(EGFR(G719C))19EGFR(G719C)Outcome
38Kd(EGFR(G719C))*19FloatμM
39Outcome(EPHA3)20EPHA3Outcome
40Kd(EPHA3)*20FloatμM
41Outcome(EPHA6)21EPHA6Outcome
42Kd(EPHA6)*21FloatμM
43Outcome(EPHA7)22EPHA7Outcome
44Kd(EPHA7)*22FloatμM
45Outcome(EPHB3)23EPHB3Outcome
46Kd(EPHB3)*23FloatμM
47Outcome(EPHB4)24EPHB4Outcome
48Kd(EPHB4)*24FloatμM
49Outcome(ERK8)25ERK8Outcome
50Kd(ERK8)*25FloatμM
51Outcome(FLT1)26FLT1Outcome
52Kd(FLT1)*26FloatμM
53Outcome(FLT3)27FLT3Outcome
54Kd(FLT3)*27FloatμM
55Outcome(FLT3(D835H))28FLT3(D835H)Outcome
56Kd(FLT3(D835H))*28FloatμM
57Outcome(FLT3(D835Y))29FLT3(D835Y)Outcome
58Kd(FLT3(D835Y))*29FloatμM
59Outcome(FLT3(ITD))30FLT3(ITD)Outcome
60Kd(FLT3(ITD))*30FloatμM
61Outcome(FLT3(N841I))31FLT3(N841I)Outcome
62Kd(FLT3(N841I))*31FloatμM
63Outcome(FLT4)32FLT4Outcome
64Kd(FLT4)*32FloatμM
65Outcome(FRK)33FRKOutcome
66Kd(FRK)*33FloatμM
67Outcome(INSRR)34INSRROutcome
68Kd(INSRR)*34FloatμM
69Outcome(JNK2)35JNK2Outcome
70Kd(JNK2)*35FloatμM
71Outcome(KIT)36KITOutcome
72Kd(KIT)*36FloatμM
73Outcome(KIT(D816V))37KIT(D816V)Outcome
74Kd(KIT(D816V))*37FloatμM
75Outcome(KIT(V559D T670I))38KIT(V559D T670I)Outcome
76Kd(KIT(V559D T670I))*38FloatμM
77Outcome(KIT(V559D V654A))39KIT(V559D V654A)Outcome
78Kd(KIT(V559D V654A))*39FloatμM
79Outcome(KIT(V559D))40KIT(V559D)Outcome
80Kd(KIT(V559D))*40FloatμM
81Outcome(LATS2)41LATS2Outcome
82Kd(LATS2)*41FloatμM
83Outcome(LIMK2)42LIMK2Outcome
84Kd(LIMK2)*42FloatμM
85Outcome(LOK)43LOKOutcome
86Kd(LOK)*43FloatμM
87Outcome(LTK)44LTKOutcome
88Kd(LTK)*44FloatμM
89Outcome(MAP4K1)45MAP4K1Outcome
90Kd(MAP4K1)*45FloatμM
91Outcome(MAP4K3)46MAP4K3Outcome
92Kd(MAP4K3)*46FloatμM
93Outcome(MAP4K5)47MAP4K5Outcome
94Kd(MAP4K5)*47FloatμM
95Outcome(MERTK)48MERTKOutcome
96Kd(MERTK)*48FloatμM
97Outcome(MET)49METOutcome
98Kd(MET)*49FloatμM
99Outcome(MKNK1)50MKNK1Outcome
100Kd(MKNK1)*50FloatμM
101Outcome(MKNK2)51MKNK2Outcome
102Kd(MKNK2)*51FloatμM
103Outcome(MST1)52MST1Outcome
104Kd(MST1)*52FloatμM
105Outcome(MST2)53MST2Outcome
106Kd(MST2)*53FloatμM
107Outcome(MUSK)54MUSKOutcome
108Kd(MUSK)*54FloatμM
109Outcome(PDGFRA)55PDGFRAOutcome
110Kd(PDGFRA)*55FloatμM
111Outcome(PDGFRB)56PDGFRBOutcome
112Kd(PDGFRB)*56FloatμM
113Outcome(PKAC-alpha)57PKAC-alphaOutcome
114Kd(PKAC-alpha)*57FloatμM
115Outcome(PLK3)58PLK3Outcome
116Kd(PLK3)*58FloatμM
117Outcome(RET)59RETOutcome
118Kd(RET)*59FloatμM
119Outcome(RET(M918T))60RET(M918T)Outcome
120Kd(RET(M918T))*60FloatμM
121Outcome(RIPK1)61RIPK1Outcome
122Kd(RIPK1)*61FloatμM
123Outcome(RPS6KA4(Kin.Dom.1 - N-terminal))62RPS6KA4(Kin.Dom.1 - N-terminal)Outcome
124Kd(RPS6KA4(Kin.Dom.1 - N-terminal))*62FloatμM
125Outcome(RPS6KA5(Kin.Dom.1 - N-terminal))63RPS6KA5(Kin.Dom.1 - N-terminal)Outcome
126Kd(RPS6KA5(Kin.Dom.1 - N-terminal))*63FloatμM
127Outcome(SLK)64SLKOutcome
128Kd(SLK)*64FloatμM
129Outcome(STK33)65STK33Outcome
130Kd(STK33)*65FloatμM
131Outcome(TIE1)66TIE1Outcome
132Kd(TIE1)*66FloatμM
133Outcome(TIE2)67TIE2Outcome
134Kd(TIE2)*67FloatμM
135Outcome(TRKA)68TRKAOutcome
136Kd(TRKA)*68FloatμM
137Outcome(TRKB)69TRKBOutcome
138Kd(TRKB)*69FloatμM
139Outcome(TRKC)70TRKCOutcome
140Kd(TRKC)*70FloatμM
141Outcome(VEGFR2)71VEGFR2Outcome
142Kd(VEGFR2)*71FloatμM
143Outcome(YANK2)72YANK2Outcome
144Kd(YANK2)*72FloatμM
145Outcome(ABL1)73ABL1Outcome
146Kd(ABL1)*73FloatμM
147Outcome(BLK)74BLKOutcome
148Kd(BLK)*74FloatμM
149Outcome(BRAF)75BRAFOutcome
150Kd(BRAF)*75FloatμM
151Outcome(BRAF(V600E))76BRAF(V600E)Outcome
152Kd(BRAF(V600E))*76FloatμM
153Outcome(CIT)77CITOutcome
154Kd(CIT)*77FloatμM
155Outcome(EGFR)78EGFROutcome
156Kd(EGFR)*78FloatμM
157Outcome(EGFR(G719S))79EGFR(G719S)Outcome
158Kd(EGFR(G719S))*79FloatμM
159Outcome(EGFR(L747-E749del A750P))80EGFR(L747-E749del A750P)Outcome
160Kd(EGFR(L747-E749del A750P))*80FloatμM
161Outcome(EGFR(L747-S752del P753S))81EGFR(L747-S752del P753S)Outcome
162Kd(EGFR(L747-S752del P753S))*81FloatμM
163Outcome(EGFR(L747-T751del Sins))82EGFR(L747-T751del Sins)Outcome
164Kd(EGFR(L747-T751del Sins))*82FloatμM
165Outcome(EGFR(L861Q))83EGFR(L861Q)Outcome
166Kd(EGFR(L861Q))*83FloatμM
167Outcome(FGFR1)84FGFR1Outcome
168Kd(FGFR1)*84FloatμM
169Outcome(FGFR4)85FGFR4Outcome
170Kd(FGFR4)*85FloatμM
171Outcome(FGR)86FGROutcome
172Kd(FGR)*86FloatμM
173Outcome(FYN)87FYNOutcome
174Kd(FYN)*87FloatμM
175Outcome(GCN2(Kin.Dom.2 S808G))88GCN2(Kin.Dom.2 S808G)Outcome
176Kd(GCN2(Kin.Dom.2 S808G))*88FloatμM
177Outcome(LCK)89LCKOutcome
178Kd(LCK)*89FloatμM
179Outcome(LYN)90LYNOutcome
180Kd(LYN)*90FloatμM
181Outcome(PTK6)91PTK6Outcome
182Kd(PTK6)*91FloatμM
183Outcome(RAF1)92RAF1Outcome
184Kd(RAF1)*92FloatμM
185Outcome(TNNI3K)93TNNI3KOutcome
186Kd(TNNI3K)*93FloatμM
187Outcome(ZAK)94ZAKOutcome
188Kd(ZAK)*94FloatμM
189Outcome(ABL1(E255K))95ABL1(E255K)Outcome
190Kd(ABL1(E255K))*95FloatμM
191Outcome(ABL1(H396P))96ABL1(H396P)Outcome
192Kd(ABL1(H396P))*96FloatμM
193Outcome(ABL1(M351T))97ABL1(M351T)Outcome
194Kd(ABL1(M351T))*97FloatμM
195Outcome(ABL1(Q252H))98ABL1(Q252H)Outcome
196Kd(ABL1(Q252H))*98FloatμM
197Outcome(ABL1(Y253F))99ABL1(Y253F)Outcome
198Kd(ABL1(Y253F))*99FloatμM
199Outcome(ABL2)100ABL2Outcome
200Kd(ABL2)*100FloatμM
201Outcome(AMPK-alpha1)101AMPK-alpha1Outcome
202Kd(AMPK-alpha1)*101FloatμM
203Outcome(ANKK1)102ANKK1Outcome
204Kd(ANKK1)*102FloatμM
205Outcome(CAMK1)103CAMK1Outcome
206Kd(CAMK1)*103FloatμM
207Outcome(CAMK4)104CAMK4Outcome
208Kd(CAMK4)*104FloatμM
209Outcome(CAMKK1)105CAMKK1Outcome
210Kd(CAMKK1)*105FloatμM
211Outcome(CAMKK2)106CAMKK2Outcome
212Kd(CAMKK2)*106FloatμM
213Outcome(CDK2)107CDK2Outcome
214Kd(CDK2)*107FloatμM
215Outcome(CDK3)108CDK3Outcome
216Kd(CDK3)*108FloatμM
217Outcome(CDK5)109CDK5Outcome
218Kd(CDK5)*109FloatμM
219Outcome(CLK2)110CLK2Outcome
220Kd(CLK2)*110FloatμM
221Outcome(CSK)111CSKOutcome
222Kd(CSK)*111FloatμM
223Outcome(CSNK1D)112CSNK1DOutcome
224Kd(CSNK1D)*112FloatμM
225Outcome(CSNK1E)113CSNK1EOutcome
226Kd(CSNK1E)*113FloatμM
227Outcome(CSNK1G2)114CSNK1G2Outcome
228Kd(CSNK1G2)*114FloatμM
229Outcome(CSNK1G3)115CSNK1G3Outcome
230Kd(CSNK1G3)*115FloatμM
231Outcome(DAPK3)116DAPK3Outcome
232Kd(DAPK3)*116FloatμM
233Outcome(DLK)117DLKOutcome
234Kd(DLK)*117FloatμM
235Outcome(EGFR(E746-A750del))118EGFR(E746-A750del)Outcome
236Kd(EGFR(E746-A750del))*118FloatμM
237Outcome(EGFR(L858R))119EGFR(L858R)Outcome
238Kd(EGFR(L858R))*119FloatμM
239Outcome(EPHA2)120EPHA2Outcome
240Kd(EPHA2)*120FloatμM
241Outcome(EPHA4)121EPHA4Outcome
242Kd(EPHA4)*121FloatμM
243Outcome(EPHA5)122EPHA5Outcome
244Kd(EPHA5)*122FloatμM
245Outcome(EPHA8)123EPHA8Outcome
246Kd(EPHA8)*123FloatμM
247Outcome(EPHB1)124EPHB1Outcome
248Kd(EPHB1)*124FloatμM
249Outcome(EPHB2)125EPHB2Outcome
250Kd(EPHB2)*125FloatμM
251Outcome(FER)126FEROutcome
252Kd(FER)*126FloatμM
253Outcome(FES)127FESOutcome
254Kd(FES)*127FloatμM
255Outcome(FGFR2)128FGFR2Outcome
256Kd(FGFR2)*128FloatμM
257Outcome(GAK)129GAKOutcome
258Kd(GAK)*129FloatμM
259Outcome(HCK)130HCKOutcome
260Kd(HCK)*130FloatμM
261Outcome(ITK)131ITKOutcome
262Kd(ITK)*131FloatμM
263Outcome(JAK2(Kin.Dom.2/JH1 - catalytic))132JAK2(Kin.Dom.2/JH1 - catalytic)Outcome
264Kd(JAK2(Kin.Dom.2/JH1 - catalytic))*132FloatμM
265Outcome(JAK3(Kin.Dom.2/JH1 - catalytic))133JAK3(Kin.Dom.2/JH1 - catalytic)Outcome
266Kd(JAK3(Kin.Dom.2/JH1 - catalytic))*133FloatμM
267Outcome(JNK1)134JNK1Outcome
268Kd(JNK1)*134FloatμM
269Outcome(JNK3)135JNK3Outcome
270Kd(JNK3)*135FloatμM
271Outcome(LATS1)136LATS1Outcome
272Kd(LATS1)*136FloatμM
273Outcome(MAP4K4)137MAP4K4Outcome
274Kd(MAP4K4)*137FloatμM
275Outcome(MELK)138MELKOutcome
276Kd(MELK)*138FloatμM
277Outcome(MYLK2)139MYLK2Outcome
278Kd(MYLK2)*139FloatμM
279Outcome(MYO3A)140MYO3AOutcome
280Kd(MYO3A)*140FloatμM
281Outcome(MYO3B)141MYO3BOutcome
282Kd(MYO3B)*141FloatμM
283Outcome(NEK5)142NEK5Outcome
284Kd(NEK5)*142FloatμM
285Outcome(NLK)143NLKOutcome
286Kd(NLK)*143FloatμM
287Outcome(PCTK1)144PCTK1Outcome
288Kd(PCTK1)*144FloatμM
289Outcome(PCTK2)145PCTK2Outcome
290Kd(PCTK2)*145FloatμM
291Outcome(PCTK3)146PCTK3Outcome
292Kd(PCTK3)*146FloatμM
293Outcome(PFTK1)147PFTK1Outcome
294Kd(PFTK1)*147FloatμM
295Outcome(PKAC-beta)148PKAC-betaOutcome
296Kd(PKAC-beta)*148FloatμM
297Outcome(PRKCQ)149PRKCQOutcome
298Kd(PRKCQ)*149FloatμM
299Outcome(PRKD1)150PRKD1Outcome
300Kd(PRKD1)*150FloatμM
301Outcome(PRKD2)151PRKD2Outcome
302Kd(PRKD2)*151FloatμM
303Outcome(PRKD3)152PRKD3Outcome
304Kd(PRKD3)*152FloatμM
305Outcome(PRKR)153PRKROutcome
306Kd(PRKR)*153FloatμM
307Outcome(PTK2B)154PTK2BOutcome
308Kd(PTK2B)*154FloatμM
309Outcome(RIPK2)155RIPK2Outcome
310Kd(RIPK2)*155FloatμM
311Outcome(ROS1)156ROS1Outcome
312Kd(ROS1)*156FloatμM
313Outcome(RPS6KA2(Kin.Dom.2 - C-terminal))157RPS6KA2(Kin.Dom.2 - C-terminal)Outcome
314Kd(RPS6KA2(Kin.Dom.2 - C-terminal))*157FloatμM
315Outcome(RPS6KA6(Kin.Dom.2 - C-terminal))158RPS6KA6(Kin.Dom.2 - C-terminal)Outcome
316Kd(RPS6KA6(Kin.Dom.2 - C-terminal))*158FloatμM
317Outcome(SNF1LK)159SNF1LKOutcome
318Kd(SNF1LK)*159FloatμM
319Outcome(SRC)160SRCOutcome
320Kd(SRC)*160FloatμM
321Outcome(SRMS)161SRMSOutcome
322Kd(SRMS)*161FloatμM
323Outcome(STK36)162STK36Outcome
324Kd(STK36)*162FloatμM
325Outcome(SYK)163SYKOutcome
326Kd(SYK)*163FloatμM
327Outcome(TESK1)164TESK1Outcome
328Kd(TESK1)*164FloatμM
329Outcome(TGFBR2)165TGFBR2Outcome
330Kd(TGFBR2)*165FloatμM
331Outcome(TNIK)166TNIKOutcome
332Kd(TNIK)*166FloatμM
333Outcome(TNK1)167TNK1Outcome
334Kd(TNK1)*167FloatμM
335Outcome(TTK)168TTKOutcome
336Kd(TTK)*168FloatμM
337Outcome(TYK2(Kin.Dom.2/JH1 - catalytic))169TYK2(Kin.Dom.2/JH1 - catalytic)Outcome
338Kd(TYK2(Kin.Dom.2/JH1 - catalytic))*169FloatμM
339Outcome(YES)170YESOutcome
340Kd(YES)*170FloatμM
341Outcome(YSK1)171YSK1Outcome
342Kd(YSK1)*171FloatμM
343Outcome(p38-alpha)172p38-alphaOutcome
344Kd(p38-alpha)*172FloatμM
345Outcome(p38-beta)173p38-betaOutcome
346Kd(p38-beta)*173FloatμM
347Outcome(p38-gamma)174p38-gammaOutcome
348Kd(p38-gamma)*174FloatμM
349Outcome(EGFR(S752-I759del))175EGFR(S752-I759del)Outcome
350Kd(EGFR(S752-I759del))*175FloatμM
351Outcome(ERBB2)176ERBB2Outcome
352Kd(ERBB2)*176FloatμM
353Outcome(ERBB4)177ERBB4Outcome
354Kd(ERBB4)*177FloatμM
355Outcome(MEK2)178MEK2Outcome
356Kd(MEK2)*178FloatμM
357Outcome(PLK4)179PLK4Outcome
358Kd(PLK4)*179FloatμM
359Outcome(DMPK2)180DMPK2Outcome
360Kd(DMPK2)*180FloatμM
361Outcome(EPHA1)181EPHA1Outcome
362Kd(EPHA1)*181FloatμM
363Outcome(MRCKA)182MRCKAOutcome
364Kd(MRCKA)*182FloatμM
365Outcome(MRCKB)183MRCKBOutcome
366Kd(MRCKB)*183FloatμM
367Outcome(PTK2)184PTK2Outcome
368Kd(PTK2)*184FloatμM
369Outcome(DCAMKL1)185DCAMKL1Outcome
370Kd(DCAMKL1)*185FloatμM
371Outcome(DCAMKL2)186DCAMKL2Outcome
372Kd(DCAMKL2)*186FloatμM
373Outcome(DCAMKL3)187DCAMKL3Outcome
374Kd(DCAMKL3)*187FloatμM
375Outcome(DRAK1)188DRAK1Outcome
376Kd(DRAK1)*188FloatμM
377Outcome(DYRK1B)189DYRK1BOutcome
378Kd(DYRK1B)*189FloatμM
379Outcome(ERK3)190ERK3Outcome
380Kd(ERK3)*190FloatμM
381Outcome(ERK4)191ERK4Outcome
382Kd(ERK4)*191FloatμM
383Outcome(ERK5)192ERK5Outcome
384Kd(ERK5)*192FloatμM
385Outcome(GSK3A)193GSK3AOutcome
386Kd(GSK3A)*193FloatμM
387Outcome(GSK3B)194GSK3BOutcome
388Kd(GSK3B)*194FloatμM
389Outcome(IRAK3)195IRAK3Outcome
390Kd(IRAK3)*195FloatμM
391Outcome(MLCK)196MLCKOutcome
392Kd(MLCK)*196FloatμM
393Outcome(PAK3)197PAK3Outcome
394Kd(PAK3)*197FloatμM
395Outcome(PHKG1)198PHKG1Outcome
396Kd(PHKG1)*198FloatμM
397Outcome(SNARK)199SNARKOutcome
398Kd(SNARK)*199FloatμM
399Outcome(AAK1)200AAK1Outcome
400Kd(AAK1)*200FloatμM
401Outcome(AMPK-alpha2)201AMPK-alpha2Outcome
402Kd(AMPK-alpha2)*201FloatμM
403Outcome(ARK5)202ARK5Outcome
404Kd(ARK5)*202FloatμM
405Outcome(BIKE)203BIKEOutcome
406Kd(BIKE)*203FloatμM
407Outcome(CHEK1)204CHEK1Outcome
408Kd(CHEK1)*204FloatμM
409Outcome(CSNK2A1)205CSNK2A1Outcome
410Kd(CSNK2A1)*205FloatμM
411Outcome(CSNK2A2)206CSNK2A2Outcome
412Kd(CSNK2A2)*206FloatμM
413Outcome(DRAK2)207DRAK2Outcome
414Kd(DRAK2)*207FloatμM
415Outcome(FGFR3)208FGFR3Outcome
416Kd(FGFR3)*208FloatμM
417Outcome(FGFR3(G697C))209FGFR3(G697C)Outcome
418Kd(FGFR3(G697C))*209FloatμM
419Outcome(IKK-epsilon)210IKK-epsilonOutcome
420Kd(IKK-epsilon)*210FloatμM
421Outcome(JAK1(Kin.Dom.1/JH2 - pseudokinase))211JAK1(Kin.Dom.1/JH2 - pseudokinase)Outcome
422Kd(JAK1(Kin.Dom.1/JH2 - pseudokinase))*211FloatμM
423Outcome(LKB1)212LKB1Outcome
424Kd(LKB1)*212FloatμM
425Outcome(MAP3K4)213MAP3K4Outcome
426Kd(MAP3K4)*213FloatμM
427Outcome(MARK1)214MARK1Outcome
428Kd(MARK1)*214FloatμM
429Outcome(MARK2)215MARK2Outcome
430Kd(MARK2)*215FloatμM
431Outcome(MARK3)216MARK3Outcome
432Kd(MARK3)*216FloatμM
433Outcome(MARK4)217MARK4Outcome
434Kd(MARK4)*217FloatμM
435Outcome(MEK1)218MEK1Outcome
436Kd(MEK1)*218FloatμM
437Outcome(MLK1)219MLK1Outcome
438Kd(MLK1)*219FloatμM
439Outcome(MLK3)220MLK3Outcome
440Kd(MLK3)*220FloatμM
441Outcome(MST3)221MST3Outcome
442Kd(MST3)*221FloatμM
443Outcome(MST4)222MST4Outcome
444Kd(MST4)*222FloatμM
445Outcome(MYLK)223MYLKOutcome
446Kd(MYLK)*223FloatμM
447Outcome(NEK2)224NEK2Outcome
448Kd(NEK2)*224FloatμM
449Outcome(NEK6)225NEK6Outcome
450Kd(NEK6)*225FloatμM
451Outcome(NEK7)226NEK7Outcome
452Kd(NEK7)*226FloatμM
453Outcome(NEK9)227NEK9Outcome
454Kd(NEK9)*227FloatμM
455Outcome(PHKG2)228PHKG2Outcome
456Kd(PHKG2)*228FloatμM
457Outcome(PIP5K1A)229PIP5K1AOutcome
458Kd(PIP5K1A)*229FloatμM
459Outcome(PIP5K2B)230PIP5K2BOutcome
460Kd(PIP5K2B)*230FloatμM
461Outcome(PKN1)231PKN1Outcome
462Kd(PKN1)*231FloatμM
463Outcome(PKN2)232PKN2Outcome
464Kd(PKN2)*232FloatμM
465Outcome(RIOK1)233RIOK1Outcome
466Kd(RIOK1)*233FloatμM
467Outcome(RIOK3)234RIOK3Outcome
468Kd(RIOK3)*234FloatμM
469Outcome(RPS6KA1(Kin.Dom.1 - N-terminal))235RPS6KA1(Kin.Dom.1 - N-terminal)Outcome
470Kd(RPS6KA1(Kin.Dom.1 - N-terminal))*235FloatμM
471Outcome(RPS6KA2(Kin.Dom.1 - N-terminal))236RPS6KA2(Kin.Dom.1 - N-terminal)Outcome
472Kd(RPS6KA2(Kin.Dom.1 - N-terminal))*236FloatμM
473Outcome(RPS6KA3(Kin.Dom.1 - N-terminal))237RPS6KA3(Kin.Dom.1 - N-terminal)Outcome
474Kd(RPS6KA3(Kin.Dom.1 - N-terminal))*237FloatμM
475Outcome(RPS6KA6(Kin.Dom.1 - N-terminal))238RPS6KA6(Kin.Dom.1 - N-terminal)Outcome
476Kd(RPS6KA6(Kin.Dom.1 - N-terminal))*238FloatμM
477Outcome(SNF1LK2)239SNF1LK2Outcome
478Kd(SNF1LK2)*239FloatμM
479Outcome(SRPK1)240SRPK1Outcome
480Kd(SRPK1)*240FloatμM
481Outcome(SRPK2)241SRPK2Outcome
482Kd(SRPK2)*241FloatμM
483Outcome(SgK085)242SgK085Outcome
484Kd(SgK085)*242FloatμM
485Outcome(TLK2)243TLK2Outcome
486Kd(TLK2)*243FloatμM
487Outcome(TYRO3)244TYRO3Outcome
488Kd(TYRO3)*244FloatμM
489Outcome(WEE1)245WEE1Outcome
490Kd(WEE1)*245FloatμM
491Outcome(ACVR1)246ACVR1Outcome
492Kd(ACVR1)*246FloatμM
493Outcome(ADCK3)247ADCK3Outcome
494Kd(ADCK3)*247FloatμM
495Outcome(ADCK4)248ADCK4Outcome
496Kd(ADCK4)*248FloatμM
497Outcome(BMX)249BMXOutcome
498Kd(BMX)*249FloatμM
499Outcome(BTK)250BTKOutcome
500Kd(BTK)*250FloatμM
501Outcome(RPS6KA1(Kin.Dom.2 - C-terminal))251RPS6KA1(Kin.Dom.2 - C-terminal)Outcome
502Kd(RPS6KA1(Kin.Dom.2 - C-terminal))*251FloatμM
503Outcome(TEC)252TECOutcome
504Kd(TEC)*252FloatμM
505Outcome(TGFBR1)253TGFBR1Outcome
506Kd(TGFBR1)*253FloatμM
507Outcome(TXK)254TXKOutcome
508Kd(TXK)*254FloatμM
509Outcome(ACVR1B)255ACVR1BOutcome
510Kd(ACVR1B)*255FloatμM
511Outcome(ACVR2A)256ACVR2AOutcome
512Kd(ACVR2A)*256FloatμM
513Outcome(ACVR2B)257ACVR2BOutcome
514Kd(ACVR2B)*257FloatμM
515Outcome(ACVRL1)258ACVRL1Outcome
516Kd(ACVRL1)*258FloatμM
517Outcome(DMPK)259DMPKOutcome
518Kd(DMPK)*259FloatμM
519Outcome(LIMK1)260LIMK1Outcome
520Kd(LIMK1)*260FloatμM
521Outcome(PKMYT1)261PKMYT1Outcome
522Kd(PKMYT1)*261FloatμM
523Outcome(TNK2)262TNK2Outcome
524Kd(TNK2)*262FloatμM
525Outcome(CAMK1D)263CAMK1DOutcome
526Kd(CAMK1D)*263FloatμM
527Outcome(CLK3)264CLK3Outcome
528Kd(CLK3)*264FloatμM
529Outcome(CSNK1A1L)265CSNK1A1LOutcome
530Kd(CSNK1A1L)*265FloatμM
531Outcome(NEK1)266NEK1Outcome
532Kd(NEK1)*266FloatμM
533Outcome(PAK1)267PAK1Outcome
534Kd(PAK1)*267FloatμM
535Outcome(PRKCD)268PRKCDOutcome
536Kd(PRKCD)*268FloatμM
537Outcome(RPS6KA4(Kin.Dom.2 - C-terminal))269RPS6KA4(Kin.Dom.2 - C-terminal)Outcome
538Kd(RPS6KA4(Kin.Dom.2 - C-terminal))*269FloatμM
539Outcome(CAMK2A)270CAMK2AOutcome
540Kd(CAMK2A)*270FloatμM
541Outcome(MLK2)271MLK2Outcome
542Kd(MLK2)*271FloatμM
543Outcome(PIM1)272PIM1Outcome
544Kd(PIM1)*272FloatμM
545Outcome(PIM2)273PIM2Outcome
546Kd(PIM2)*273FloatμM
547Outcome(PIM3)274PIM3Outcome
548Kd(PIM3)*274FloatμM
549Outcome(PRKCE)275PRKCEOutcome
550Kd(PRKCE)*275FloatμM
551Outcome(PRKCH)276PRKCHOutcome
552Kd(PRKCH)*276FloatμM
553Outcome(CAMK1G)277CAMK1GOutcome
554Kd(CAMK1G)*277FloatμM
555Outcome(MEK4)278MEK4Outcome
556Kd(MEK4)*278FloatμM
557Outcome(MEK6)279MEK6Outcome
558Kd(MEK6)*279FloatμM
559Outcome(STK16)280STK16Outcome
560Kd(STK16)*280FloatμM
561Outcome(BRSK1)281BRSK1Outcome
562Kd(BRSK1)*281FloatμM
563Outcome(BRSK2)282BRSK2Outcome
564Kd(BRSK2)*282FloatμM
565Outcome(CSNK1G1)283CSNK1G1Outcome
566Kd(CSNK1G1)*283FloatμM
567Outcome(MEK3)284MEK3Outcome
568Kd(MEK3)*284FloatμM
569Outcome(PAK4)285PAK4Outcome
570Kd(PAK4)*285FloatμM
571Outcome(PAK6)286PAK6Outcome
572Kd(PAK6)*286FloatμM
573Outcome(PAK7/PAK5)287PAK7/PAK5Outcome
574Kd(PAK7/PAK5)*287FloatμM
575Outcome(PDPK1)288PDPK1Outcome
576Kd(PDPK1)*288FloatμM
577Outcome(PLK1)289PLK1Outcome
578Kd(PLK1)*289FloatμM
579Outcome(TLK1)290TLK1Outcome
580Kd(TLK1)*290FloatμM
581Outcome(AKT3)291AKT3Outcome
582Kd(AKT3)*291FloatμM
583Outcome(CAMK2D)292CAMK2DOutcome
584Kd(CAMK2D)*292FloatμM
585Outcome(CAMK2G)293CAMK2GOutcome
586Kd(CAMK2G)*293FloatμM
587Outcome(DAPK1)294DAPK1Outcome
588Kd(DAPK1)*294FloatμM
589Outcome(PRKG2)295PRKG2Outcome
590Kd(PRKG2)*295FloatμM
591Outcome(DAPK2)296DAPK2Outcome
592Kd(DAPK2)*296FloatμM
593Outcome(PIK3CA)297PIK3CAOutcome
594Kd(PIK3CA)*297FloatμM
595Outcome(PIK3CA(E545K))298PIK3CA(E545K)Outcome
596Kd(PIK3CA(E545K))*298FloatμM
597Outcome(AKT1)299AKT1Outcome
598Kd(AKT1)*299FloatμM
599Outcome(AKT2)300AKT2Outcome
600Kd(AKT2)*300FloatμM
601Outcome(CAMK2B)301CAMK2BOutcome
602Kd(CAMK2B)*301FloatμM
603Outcome(PAK2)302PAK2Outcome
604Kd(PAK2)*302FloatμM
605Outcome(PRKG1)303PRKG1Outcome
606Kd(PRKG1)*303FloatμM
607Outcome(PRKX)304PRKXOutcome
608Kd(PRKX)*304FloatμM
609Outcome(TSSK1)305TSSK1Outcome
610Kd(TSSK1)*305FloatμM
611Outcome(ZAP70)306ZAP70Outcome
612Kd(ZAP70)*306FloatμM
613Outcome(INSR)307INSROutcome
614Kd(INSR)*307FloatμM
615Outcome(NDR2)308NDR2Outcome
616Kd(NDR2)*308FloatμM
617Outcome(RPS6KA5(Kin.Dom.2 - C-terminal))309RPS6KA5(Kin.Dom.2 - C-terminal)Outcome
618Kd(RPS6KA5(Kin.Dom.2 - C-terminal))*309FloatμM
619Outcome(BMPR1A)310BMPR1AOutcome
620Kd(BMPR1A)*310FloatμM
621Outcome(ERK1)311ERK1Outcome
622Kd(ERK1)*311FloatμM
623Outcome(ERK2)312ERK2Outcome
624Kd(ERK2)*312FloatμM
625Outcome(IGF1R)313IGF1ROutcome
626Kd(IGF1R)*313FloatμM
627Outcome(MAP3K5)314MAP3K5Outcome
628Kd(MAP3K5)*314FloatμM
629Outcome(MAPKAPK2)315MAPKAPK2Outcome
630Kd(MAPKAPK2)*315FloatμM
631Outcome(YANK3)316YANK3Outcome
632Kd(YANK3)*316FloatμM
* Activity Concentration. § Panel component ID.

Classification
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