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BioAssay: AID 1085724

Displacement of [3H]estradiol from full-length Homo sapiens (human) ERalpha relative to estradiol

Displacement of [3H]estradiol from full-length Homo sapiens (human) ERalpha relative to estradiol ..more
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 Tested Compounds
 Tested Compounds
All(30)
 
 
Unspecified(30)
 
 
 Tested Substances
 Tested Substances
All(30)
 
 
Unspecified(30)
 
 
 Related BioAssays
 Related BioAssays
AID: 1085724
Data Source: ChEMBL (902275)
Depositor Category: Literature, Extracted
Deposit Date: 2014-08-26
Modify Date: 2014-12-06

Data Table ( Complete ):           View All Data
Target
Sequence: RecName: Full=Estrogen receptor; Short=ER; AltName: Full=ER-alpha; AltName: Full=Estradiol receptor; AltName: Full=Nuclear receptor subfamily 3 group A member 1
Description ..   
Protein Family: Ligand binding domain of Estrogen receptor, which are activated by the hormone 17beta-estradiol (estrogen)
Comment ..   

Gene:ESR1     Related Protein 3D Structures     More BioActivity Data..
Tested Compounds:
Description:
Displacement of [3H]estradiol from full-length Homo sapiens (human) ERalpha relative to estradiol
Comment
Publication:
Journal: Med Chem Res
Year: 2012
Volume: 21
Issue: 9
First Page: 2652
Last Page: 2660
Categorized Comment - additional comments and annotations
From BioAssay Depositor:
Assay Type: Binding
Target Type: Target is a single protein chain
Assay Data Source: Scientific Literature
Result Definitions
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1RBA activity commentRBA activity commentString
2RBA standard flagRBA standard flagInteger
3RBA qualifierRBA qualifierString
4RBA published valueRBA published valueFloat%
5RBA standard valueRBA standard valueFloat%

Data Table (Concise)
Data Table ( Complete ):     View All Data
Classification
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